C6–H Bond Functionalization of Indoles: A New Gate DOI
Nurullah Saraçoğlu, Yunus Taskesenligil

Synthesis, Journal Year: 2023, Volume and Issue: 55(21), P. 3417 - 3433

Published: March 8, 2023

Abstract Indoles are valuable precursors in medicinal, bioorganic, and material chemistry particularly serve as a platform for diversity. However, the scope of C6-functionalization indoles was limited until recently. In this short review, we summarize developments reactions involving transition-metal-catalyzed functionalization Brønsted Lewis acid catalyzed processes. The regioselectivity is controlled by remote-C–H activation hydrogen bond formation. 1 Introduction 2 Transition-Metal-Catalyzed Functionalization 3 Acid-Catalyzed Processes 4 Conclusion

Language: Английский

1,6-Conjugate addition of in situ generated aryldiazenes to p-quinone methides DOI

Ajay G. Mamale,

Sayantan Paul,

Rajesh G. Gonnade

et al.

Organic & Biomolecular Chemistry, Journal Year: 2024, Volume and Issue: 22(27), P. 5636 - 5645

Published: Jan. 1, 2024

Herein we report a transition-metal free, base-mediated 1,6-conjugate addition of aryldiazenes to para -quinone methides ( p -QMs).

Language: Английский

Citations

3

Solvent Dictated Organic Transformations DOI
Tamanna Khandelia, Pritishree Panigrahi, Subhendu Ghosh

et al.

Chemistry - An Asian Journal, Journal Year: 2024, Volume and Issue: unknown

Published: Nov. 7, 2024

Solvent plays an important role in many chemical reactions. The C-H activation has been one of the most powerful tools organic synthesis. These reactions are often assisted by solvents which not only provide a medium for but also facilitate reaching to product stage. solvent helps reaction profile both chemically and energetically reach targeted product. Organic transformations via from assistance perspective discussed this review. Various such as tetrahydrofuran (THF), MeCN, dichloromethane (DCM), dimethoxyethane (DME), 1,2-dichloroethane (1,2-DCE), dimethylformamide (DMF), dimethylsulfoxide (DMSO), isopropyl nitrile (

Language: Английский

Citations

1

C6–H Bond Functionalization of Indoles: A New Gate DOI
Nurullah Saraçoğlu, Yunus Taskesenligil

Synthesis, Journal Year: 2023, Volume and Issue: 55(21), P. 3417 - 3433

Published: March 8, 2023

Abstract Indoles are valuable precursors in medicinal, bioorganic, and material chemistry particularly serve as a platform for diversity. However, the scope of C6-functionalization indoles was limited until recently. In this short review, we summarize developments reactions involving transition-metal-catalyzed functionalization Brønsted Lewis acid catalyzed processes. The regioselectivity is controlled by remote-C–H activation hydrogen bond formation. 1 Introduction 2 Transition-Metal-Catalyzed Functionalization 3 Acid-Catalyzed Processes 4 Conclusion

Language: Английский

Citations

1