ChemistrySelect, Journal Year: 2024, Volume and Issue: 9(35)
Published: Sept. 13, 2024
Abstract Primary alcohols 2(a–h) and o‐aminobenzamides 1(a–h) can be selectively oxidized electrochemically to yield dihydroquinazolinone 4(a–h) quinazolinones 5(a–h) in an efficient chemoselective manner. This methodology employs sodium chloride (NaCl) 3(a) as a co‐catalyst electricity the oxidizing agent, utilizing cost‐effective commercially available materials such Graphite anode, Iron (Fe) cathode, isopropyl alcohol (iPrOH) solvent weak base. The synthesis yields various quinazolinone derivatives with diverse structural characteristics good quantities, showcasing method‘s broad applicability. approach facilitates production of range dihydroquinazolinones (24 examples), highlighting its versatility compatibility different functional groups. Characterization synthesized included CHN analysis, 1 HNMR spectroscopy, determination melting points.
Language: Английский