Recent advances in therapeutic use of transforming growth factor-beta inhibitors in cancer and fibrosis DOI Creative Commons
Jing He, Yan Gao, Linyuan Jing

et al.

Frontiers in Oncology, Journal Year: 2025, Volume and Issue: 15

Published: April 25, 2025

Transforming growth factor-beta (TGF-β) has long been known to be associated with early embryonic development and organogenesis, immune supervision, tissue repair homeostasis in adults. TGF-β complex roles fibrosis cancer that may opposing at different stages of these diseases. Under pathological conditions, overexpression causes epithelial–mesenchymal transition, deposition extracellular matrix, formation cancer-associated fibroblasts, leading fibrotic disease or cancer. Fibroblasts, epithelial cells, cells are the most common targets TGF-β, while TGF-β-associated Given critical role its downstream molecules progression cancer, therapies targeting signaling appear a promising strategy. Preclinical clinical studies have investigated including antisense oligonucleotides, monoclonal antibodies, ligand traps. However, targeted therapy hindered by systemic cytotoxicity. This review discusses molecular mechanisms highlights for as therapeutic strategy related

Language: Английский

Reprogramming the breast tumor immune microenvironment: cold-to-hot transition for enhanced immunotherapy DOI Creative Commons
Saber Imani, Reyhaneh Farghadani, Ghazaal Roozitalab

et al.

Journal of Experimental & Clinical Cancer Research, Journal Year: 2025, Volume and Issue: 44(1)

Published: April 25, 2025

Abstract This review discusses reprogramming the breast tumor immune microenvironment from an immunosuppressive cold state to immunologically active hot state. A complex interplay is revealed, in which accumulation of metabolic byproducts—such as lactate, reactive oxygen species (ROS), and ammonia—is shown impair T-cell function promote escape. It demonstrated that (TME) dominated by cytokines, including interleukin-10 (IL-10), transforming growth factorβ (TGFβ), IL-35. Notably, IL-35 produced regulatory T cells cancer cells. The conversion conventional into IL-35-producing induced cells, along with inhibition pro-inflammatory cytokine secretion, contributes suppression anti-tumor immunity. further key checkpoint molecules—such PD-1, PDL1, CTLA-4, TIM-3, LAG-3, TIGIT—are upregulated within TME, leading Tcell exhaustion diminished responses. blockade these checkpoints restore functionality proposed a strategy convert tumors ones robust effector cell infiltration. therapeutic potential chimeric antigen receptor (CAR)T therapy also explored, targeting specific tumor-associated antigens, such glycoproteins tyrosine kinases, highlighted. suggested CART efficacy can be enhanced combining inhibitors other immunomodulatory agents, thereby overcoming barriers imposed TME. Moreover, role microbiome regulating estrogen metabolism systemic inflammation reviewed. Alterations gut microbiota are affect microbiome-based interventions additional means facilitate cold-to-hot transition. concluded immunological pathways underpin suppression—through combination strategies involving blockade, therapies, modulation—the TME achieved. anticipated enhance infiltration function, improving overall immunotherapies better clinical outcomes for patients.

Language: Английский

Citations

0

Recent advances in therapeutic use of transforming growth factor-beta inhibitors in cancer and fibrosis DOI Creative Commons
Jing He, Yan Gao, Linyuan Jing

et al.

Frontiers in Oncology, Journal Year: 2025, Volume and Issue: 15

Published: April 25, 2025

Transforming growth factor-beta (TGF-β) has long been known to be associated with early embryonic development and organogenesis, immune supervision, tissue repair homeostasis in adults. TGF-β complex roles fibrosis cancer that may opposing at different stages of these diseases. Under pathological conditions, overexpression causes epithelial–mesenchymal transition, deposition extracellular matrix, formation cancer-associated fibroblasts, leading fibrotic disease or cancer. Fibroblasts, epithelial cells, cells are the most common targets TGF-β, while TGF-β-associated Given critical role its downstream molecules progression cancer, therapies targeting signaling appear a promising strategy. Preclinical clinical studies have investigated including antisense oligonucleotides, monoclonal antibodies, ligand traps. However, targeted therapy hindered by systemic cytotoxicity. This review discusses molecular mechanisms highlights for as therapeutic strategy related

Language: Английский

Citations

0