Melatonin augments anti-tumor activity and alleviates nephrotoxicity of gemcitabine in a pancreatic cancer xenograft model targeting P62/Keap1 pathway DOI Creative Commons
Samar Ibrahim,

Eman H. Yousef,

Ahmed M. El‐Dessouki

et al.

Naunyn-Schmiedeberg s Archives of Pharmacology, Journal Year: 2025, Volume and Issue: unknown

Published: March 18, 2025

Abstract Although gemcitabine is a primary chemotherapy for pancreatic cancer, its effectiveness limited by chemoresistance and nephrotoxicity, posing significant clinical challenges. Therefore, the development of novel therapeutic approaches to prevent malignancy remains crucial. This study aimed investigate potential melatonin in enhancing gemcitabine’s anticancer efficacy while mitigating nephrotoxic effects through modulation Keap1/p62 pathway. A cancer xenograft model was established rats, which received either (50 mg/kg, I.P.), or their combination three times per week 2 weeks. Our findings demonstrate that potentiates cancer-suppressing via Kelch-like-ECH associated protein-1 (Keap1)/p62 pathway, resulting reduced fibrosis, oxidative stress, inflammatory markers. Additionally, significantly mitigated gemcitabine-induced nephrotoxicity. These results suggest may serve as an adjuvant therapy treatment, reducing adverse effects.

Language: Английский

The Effect of Melatonin on Sleep Quality and Daytime Sleepiness in Parkinson’s Disease: A Systematic Review and Meta-analysis of Randomized Placebo-Controlled Trials DOI

Azzam Zrineh,

Rami Akwan,

Marwa Elsharkawy

et al.

Sleep Medicine, Journal Year: 2025, Volume and Issue: unknown, P. 106540 - 106540

Published: April 1, 2025

Language: Английский

Citations

0

The role of melatonin in the regulation of the immune system and reproductive health: mechanisms and prospects for clinical application DOI Creative Commons
M. M. Zhelavskyi, S. P. Kernychnyi, O. Ya. Dmytriv

et al.

Ukrainian Journal of Veterinary and Agricultural Sciences, Journal Year: 2025, Volume and Issue: 8(1), P. 49 - 61

Published: April 23, 2025

Melatonin is a multifunctional hormone with diverse physiological roles, particularly in immune regulation and reproductive health. While primarily synthesized by the pineal gland response to circadian rhythm, melatonin also produced extrapineal tissues such as placenta, gastrointestinal tract, organs, highlighting its systemic significance. Beyond role sleep-wake cycle regulation, exhibits potent antioxidant, anti-inflammatory, immunomodulatory properties, making it essential for maintaining cellular homeostasis overall stability. In system, contributes both innate adaptive immunity modulating cytokine production, reducing oxidative stress, enhancing cell activity. It plays protective against infections inflammatory diseases suppressing pro-inflammatory mediators interleukin-6 (IL-6) tumor necrosis factor-alpha (TNF-α) while promoting anti-inflammatory cytokines like interleukin-10 (IL-10). Additionally, influences tolerance, which critical preventing autoimmune responses ensuring successful pregnancy. females, improves oocyte quality, embryo development, pregnancy outcomes protecting ovarian follicles from damage, regulating steroidogenesis, supporting placental function. Its fetal development significant, maternal-fetal signaling, vascularization, epigenetic modifications that influence gene expression. men, spermatogenesis sperm quality boosting mitochondrial activity, decreasing safeguarding DNA damage. helps regulate production testes, optimal Given pleiotropic effects, holds substantial therapeutic potential addressing dysfunction, disorders, complications. Future research should focus on clinical applications of supplementation treating infertility, pregnancy-related complications, immune-mediated diseases. Understanding intricate relationship between melatonin, immunity, reproduction may pave way innovative strategies human veterinary medicine. roles well-known function rhythm exerts effects. function, thereby offering protection disorders. reproduction, key processes maturation, maintenance. supports fertility improving gonadotropin secretion, melatonin's involvement highlights significance gestation. widespread presents promising immune-related exploring lead novel success resilience

Language: Английский

Citations

0

Melatonin from Plants: Going Beyond Traditional Central Nervous System Targeting—A Comprehensive Review of Its Unusual Health Benefits DOI Creative Commons
Lucas Fornari Laurindo,

Otávio Augusto Garcia Simili,

Adriano Cressoni Araújo

et al.

Biology, Journal Year: 2025, Volume and Issue: 14(2), P. 143 - 143

Published: Jan. 30, 2025

Melatonin is indispensable for the homeostasis of plants and animals. In humans, it can help prevent or be an adjuvant treatment several diseases mainly related to immune system, inflammation, oxidative stress. Moreover, a melatonin-rich diet linked health benefits, such as regulation circadian rhythm, immunological epilepsy control, delaying aging process, diminishing hormones cancer. This review aimed show effects melatonin in beyond its traditional use. The results showed present scavenging free radicals, reducing inflammatory cytokines, modulating system. improve insulin resistance, blood pressure, LDL-c, adipose tissue mass, adhesion molecules, endothelial impairment, plaque formation. These result neuro- cardioprotection, improvement liver diseases, rheumatoid arthritis, dermatitis, COVID-19, polycystic ovaries, sepsis. We conclude that plant benefit patients with many besides sleep problems neurodegeneration. Plant may more cost-effective fewer adverse events than synthetic. However, clinical trials should performed adequate doses, formulation, time.

Language: Английский

Citations

0

Melatonin augments anti-tumor activity and alleviates nephrotoxicity of gemcitabine in a pancreatic cancer xenograft model targeting P62/Keap1 pathway DOI Creative Commons
Samar Ibrahim,

Eman H. Yousef,

Ahmed M. El‐Dessouki

et al.

Naunyn-Schmiedeberg s Archives of Pharmacology, Journal Year: 2025, Volume and Issue: unknown

Published: March 18, 2025

Abstract Although gemcitabine is a primary chemotherapy for pancreatic cancer, its effectiveness limited by chemoresistance and nephrotoxicity, posing significant clinical challenges. Therefore, the development of novel therapeutic approaches to prevent malignancy remains crucial. This study aimed investigate potential melatonin in enhancing gemcitabine’s anticancer efficacy while mitigating nephrotoxic effects through modulation Keap1/p62 pathway. A cancer xenograft model was established rats, which received either (50 mg/kg, I.P.), or their combination three times per week 2 weeks. Our findings demonstrate that potentiates cancer-suppressing via Kelch-like-ECH associated protein-1 (Keap1)/p62 pathway, resulting reduced fibrosis, oxidative stress, inflammatory markers. Additionally, significantly mitigated gemcitabine-induced nephrotoxicity. These results suggest may serve as an adjuvant therapy treatment, reducing adverse effects.

Language: Английский

Citations

0