Exploring Next-Generation Therapeutics: Morphic Mixtures and Specified Salts for the Treatment of Mental Disorders and CNS Modulation DOI Open Access
Robert B. Kargbo

ACS Medicinal Chemistry Letters, Journal Year: 2023, Volume and Issue: 14(9), P. 1159 - 1161

Published: Aug. 22, 2023

This Patent Highlight delves into the potential of next-generation therapeutics for treating mental disorders and modulating central nervous system (CNS). Among serotonin receptor subtypes, 5-HT2A, 5-HT2C, 5-HT1A, 5-HT1B have shown promise in CNS disorder treatment. Approved drugs targeting these receptors, such as antipsychotics psychedelics, provide valuable insights their therapeutic effects. However, modulation receptors can lead to side effects like hallucinations altered perception. The development 5-HT2A agonists with minimized mood changes improved benefits is crucial. Furthermore, exploring morphic salt mixtures specified salts offers innovative approaches effectively activity disorders.

Language: Английский

Substance use and spine density: a systematic review and meta-analysis of preclinical studies DOI
Henrique Nunes Pereira Oliva, Tiago Paiva Prudente, Eric J. Nunes

et al.

Molecular Psychiatry, Journal Year: 2024, Volume and Issue: unknown

Published: April 2, 2024

Language: Английский

Citations

4

Harnessing neuroplasticity with psychoplastogens: the essential role of psychotherapy in psychedelic treatment optimization DOI Creative Commons
Jennifer Jones

Frontiers in Psychiatry, Journal Year: 2025, Volume and Issue: 16

Published: April 8, 2025

Language: Английский

Citations

0

Effects of psychedelics on opioid use disorder: a scoping review of preclinical studies DOI Creative Commons
Alejandra Pulido-Saavedra, Henrique Nunes Pereira Oliva, Tiago Paiva Prudente

et al.

Cellular and Molecular Life Sciences, Journal Year: 2025, Volume and Issue: 82(1)

Published: Jan. 21, 2025

The current opioid crisis has had an unprecedented public health impact. Approved medications for use disorder (OUD) exist, yet their limitations indicate a need innovative treatments. Limited preliminary clinical studies suggest specific psychedelics might aid OUD treatment, though most evidence remains observational, with few controlled trials. This review aims to bridge the gap between preclinical findings and potential applications, following PRISMA-ScR guidelines. Searches included MEDLINE, Embase, Scopus, Web of Science, focusing on in vivo involving opioids animals, excluding pain those lacking control groups. Forty met criteria, covering both classic non-classic psychedelics. Most showed that 18-methoxycoronaridine (18-MC), ibogaine, noribogaine, ketamine could reduce self-administration, alleviate withdrawal symptoms, change conditioned place preference. However, seven (two 2,5-dimethoxy-4-methylamphetamine (DOM), three one 18-MC, ketamine) no improvement over controls. A methodological quality assessment rated as having unclear quality. Interestingly, are limited iboga derivatives, which were effective, but these agents may have higher cardiovascular risk than other under-explored date. strengthens support translational testing targets OUD. It also suggests include broader range beyond derivatives can explore several ongoing questions field, such mechanism action behind therapeutic effect, safety profiles, doses, frequency administrations needed.

Language: Английский

Citations

0

Gastrodin prevents stress-induced synaptic plasticity impairment and behavioral dysfunction via cAMP/PKA/CREB signaling pathway DOI

Zhihuang Zhao,

Pei Liu,

Haili Zhang

et al.

Phytomedicine, Journal Year: 2025, Volume and Issue: unknown, P. 156661 - 156661

Published: March 1, 2025

Language: Английский

Citations

0

Icariin rescues developmental BPA exposure induced spatial memory deficits in rats DOI
Danyang Li,

Shu Ai,

Chengqing Huang

et al.

Toxicology and Applied Pharmacology, Journal Year: 2023, Volume and Issue: 482, P. 116776 - 116776

Published: Dec. 1, 2023

Language: Английский

Citations

2

Exploring Next-Generation Therapeutics: Morphic Mixtures and Specified Salts for the Treatment of Mental Disorders and CNS Modulation DOI Open Access
Robert B. Kargbo

ACS Medicinal Chemistry Letters, Journal Year: 2023, Volume and Issue: 14(9), P. 1159 - 1161

Published: Aug. 22, 2023

This Patent Highlight delves into the potential of next-generation therapeutics for treating mental disorders and modulating central nervous system (CNS). Among serotonin receptor subtypes, 5-HT2A, 5-HT2C, 5-HT1A, 5-HT1B have shown promise in CNS disorder treatment. Approved drugs targeting these receptors, such as antipsychotics psychedelics, provide valuable insights their therapeutic effects. However, modulation receptors can lead to side effects like hallucinations altered perception. The development 5-HT2A agonists with minimized mood changes improved benefits is crucial. Furthermore, exploring morphic salt mixtures specified salts offers innovative approaches effectively activity disorders.

Language: Английский

Citations

0