None DOI Open Access

Oluwaseye A. Adebajo,

J. Ojo,

Perpetual K. Adebajo

et al.

International Journal of Pharmaceutical Sciences and Research, Journal Year: 2024, Volume and Issue: 15(5)

Published: May 1, 2024

Testicular toxicity has been associated with long-term paracetamol usage.Moringa oleifera is known to eliminate toxins from organs and restore functionality.This study seeks ascertain the potency of moringa in ameliorating paracetamol-induced testicular toxicity.Forty nine (49) Sprague-Dawley rats were randomly assigned into seven (7) groups composed 7 each treated for 5 weeks.One group served as control, while 3 other administered graded doses paracetamol, then 1600mg/kg extracts simultaneously.The animals sacrificed 24 hours after administration last dose using anaesthesia.The testes epididymis harvested, blood was obtained via ocular puncture.The extract mitigated dose-dependent decrease sperm count morphology.Paracetamol on hormonal milieu suppressed by treatment, yielding values closer those control group.The treatment controlled oxidative stress biomarkers their not variant when compared only.Hypospermatogenesis along restoration normal seminiferous tubules interstitial spaces observed paracetamolinduced indicates ameliorative histological effect toxicity.Therefore, use therapy reverses damaging effects testis male fertility. INTRODUCTION:A common drug used both an analgesic antipyretic 1, 2 .Paracetamol (acetaminophen) most popular non-steroidal anti-inflammatory (NSAID) available over-the-counter utilized acute chronic pain numerous clinical conditions 3, 4 .

Language: Английский

Irvingia gabonensis baill. (African Mango): A comprehensive review of its ethnopharmacological significance, unveiling its long-standing history and therapeutic potential DOI

Yassmin Raafat Hassan,

Riham A. El‐Shiekh, Hala M. El-Hefnawy

et al.

Journal of Ethnopharmacology, Journal Year: 2024, Volume and Issue: 326, P. 117942 - 117942

Published: Feb. 21, 2024

Language: Английский

Citations

5

Advancing Profiling of Secondary Antioxidant Metabolites in Allium cepa PDO Leaf Extract: Online Comprehensive Two-Dimensional Liquid Chromatography with High-Resolution Mass Spectrometry and Pre-Column DPPH Assay DOI
Giovanna Aquino, Eduardo Sommella, Emanuela Salviati

et al.

Journal of Chromatography A, Journal Year: 2025, Volume and Issue: unknown, P. 465877 - 465877

Published: March 1, 2025

Language: Английский

Citations

0

Exploring the anti-anaphylaxis potential of natural products: A Review DOI Creative Commons
Ahmed Salem Eid,

Eman M. Zaki,

Manal M. Sabry

et al.

Inflammopharmacology, Journal Year: 2025, Volume and Issue: unknown

Published: March 19, 2025

Abstract Allergies are a common health issue affecting many people around the world, especially in developed countries. They occur when immune system overreacts to substances that usually harmless. Some allergic conditions include asthma, sinus infections, skin rashes, food allergies, hay fever, severe reactions, eczema, swelling, and reactions medications or insect stings. The causes of these allergies complex often linked genetics, which can lead heightened responses known as atopy. Throughout history, plant extracts have been used for various purposes, including medicine food. In addition, their bioactive compounds show wide range beneficial effects, such reducing fighting oxidative stress, mast cell stabilizers, lowering inflammation, highlighting potential treating conditions. Flavonoids phenolic commonly anaphylaxis potent anti-inflammatory action. This review aims promote use natural products treatments anaphylaxis. discovery new drugs derived from sources holds significant promise management

Language: Английский

Citations

0

Investigating the effect of polymerase inhibitors on cellular proliferation: Computational studies, cytotoxicity, CDK1 inhibitory potential, and LC‐MS/MS cancer cell entrapment assays DOI
Faten Farouk, Ibrahim M. Ibrahim,

Salma Sherif

et al.

Chemical Biology & Drug Design, Journal Year: 2024, Volume and Issue: 103(3)

Published: March 1, 2024

Abstract Directly acting antivirals (DAAs) are a breakthrough in the treatment of HCV. There controversial reports on their tendency to induce hepatocellular carcinoma (HCC) HCV patients. Numerous have concluded that HCC is attributed patient‐related factors while others inclined attribute this as DAA side‐effect. This study aims investigate effect polymerase inhibitor DAAs, especially daclatasivir (DLT) cellular proliferation compared ribavirin (RBV). The interaction DAAs with variable cell‐cycle proteins was studied silico. binding affinities multiple targets were investigated and molecular dynamics assessed. vitro selected candidate DLT cancer cell determined CDK1 inhibitory potential evaluated. Finally, entrapment candidates assessed by an in‐house developed validated LC‐MS/MS method. results indicated antiviral agents, DLT, may exert anti‐proliferative against lines. showed be achieved via targets, including CDK1, resulting halting proliferation. exhibited remarkable permeability liver line which permits adequate targets. In conclusion, reveal cells. These pose therapeutic choice for patients suffering from liable development.

Language: Английский

Citations

2

Interactions between grapefruit juice and psychotropic medications: an update of the literature and an original case series DOI
Marcin Siwek, Anna Julia Krupa, Jarosław Woroń

et al.

Expert Opinion on Drug Metabolism & Toxicology, Journal Year: 2024, Volume and Issue: 20(5), P. 333 - 345

Published: May 3, 2024

There is a large body of preclinical data implicating that grapefruit juice (GJ) inhibits many CYP 450 isoforms. The potential GJ-to-drug high relevance to clinical psychiatry, because wide range psychotropic medicines undergo metabolism and P-gp transport.

Language: Английский

Citations

1

Phytochemical analysis and wound healing properties of Malva parviflora L. ethanolic extract DOI
Munir Ahmad Anwar,

Rania A. El Gedaily,

Abeer Salama

et al.

Journal of Ethnopharmacology, Journal Year: 2024, Volume and Issue: 337, P. 118983 - 118983

Published: Oct. 28, 2024

Language: Английский

Citations

1

A Comparative GC/MS Analysis of Citrus Essential Oils: Unveiling the Potential Benefits of Herb‐Drug Interactions in Preventing Paracetamol‐Induced Hepatotoxicity DOI Open Access
Aya S. Shalaby, Hanaa H. Eid, Riham A. El‐Shiekh

et al.

Chemistry & Biodiversity, Journal Year: 2023, Volume and Issue: 20(9)

Published: Aug. 21, 2023

Our study aimed to test the potential of Citrus oils in protecting against paracetamol (PAR)-induced hepatotoxicity. The essential Pineapple sweet orange (OO), Murcott mandarin (MO), Red grapefruit (GO), and Oval kumquat (KO) were investigated using gas chromatography coupled with mass spectrometry (GC/MS). Twenty-seven compounds identified, monoterpene hydrocarbons being abundant class. d-Limonene had highest percentage (92.98 %, 92.82 89.75 94.46 % OO, MO, GO, KO, respectively). Hierarchical cluster analysis (HCA) principal components (PCA) revealed that octanal, linalool, germacrene D, d-limonene discriminatory metabolites segregated samples into three distinct clusters. In vitro antioxidant capacities ranged from 1.2-12.27, 1.79-5.91, 235.05-585.28 μM Trolox eq/mg oil for 2,2'-azinobis(3-ethylbenzothiazoline-6-sulfonic (ABTS), ferric-reducing power (FRAP), oxygen radical absorbance capacity (ORAC), respectively. vivo, citrus exhibited a significant reduction alanine transaminase (ALT), aspartate (AST), alkaline phosphatase (ALP), nitric oxide (NO). Additionally, there was an increase glutathione reductase (GSH), liver architecture nearly normal. Molecular docking good inhibitory interaction cytochrome P450 (CYP450) isoforms 1A2, 3A4, 2E1, binding energies -6.17, -4.51, -5.61 kcal/mol,

Language: Английский

Citations

3

None DOI Open Access

Oluwaseye A. Adebajo,

J. Ojo,

Perpetual K. Adebajo

et al.

International Journal of Pharmaceutical Sciences and Research, Journal Year: 2024, Volume and Issue: 15(5)

Published: May 1, 2024

Testicular toxicity has been associated with long-term paracetamol usage.Moringa oleifera is known to eliminate toxins from organs and restore functionality.This study seeks ascertain the potency of moringa in ameliorating paracetamol-induced testicular toxicity.Forty nine (49) Sprague-Dawley rats were randomly assigned into seven (7) groups composed 7 each treated for 5 weeks.One group served as control, while 3 other administered graded doses paracetamol, then 1600mg/kg extracts simultaneously.The animals sacrificed 24 hours after administration last dose using anaesthesia.The testes epididymis harvested, blood was obtained via ocular puncture.The extract mitigated dose-dependent decrease sperm count morphology.Paracetamol on hormonal milieu suppressed by treatment, yielding values closer those control group.The treatment controlled oxidative stress biomarkers their not variant when compared only.Hypospermatogenesis along restoration normal seminiferous tubules interstitial spaces observed paracetamolinduced indicates ameliorative histological effect toxicity.Therefore, use therapy reverses damaging effects testis male fertility. INTRODUCTION:A common drug used both an analgesic antipyretic 1, 2 .Paracetamol (acetaminophen) most popular non-steroidal anti-inflammatory (NSAID) available over-the-counter utilized acute chronic pain numerous clinical conditions 3, 4 .

Language: Английский

Citations

0