Exploring the Mechanism of β-Cyclodextrin-Encased Phenolic Acids Functionalized with TPP for Antioxidant Activity and Targeting DOI Creative Commons
Christopher Sbarbaro, Valeria Márquez‐Miranda, Matías Leal

et al.

Antioxidants, Journal Year: 2025, Volume and Issue: 14(4), P. 465 - 465

Published: April 13, 2025

Oxidative stress on the mitochondria in a human cell is attributed to several life-risking conditions, and as such, importance of molecular structures packed with antioxidant properties structural characteristics enter help prevent such has been substantially relevant recent years. In this study, we investigated triphenylphosphonium (TPP)-conjugated phenolic acids encapsulated β-cyclodextrin (β-CD). We synthesized TPP conjugates caffeic, coumaric, cinnamic formed inclusion complexes β-CD. Our results showed successful encapsulation β-CD high efficiency. The maintained activity, slight reductions observed complexes. Furthermore, viability studies low cytotoxicity dds. Computational analyses revealed that conjugation preserved chemical reactivity acids. Molecular dynamics simulations demonstrated stable free energy calculations indicated significantly enhanced ability caffeic acid translocate across mitochondrial membranes. These highlight potential TPP-conjugated effective antioxidants improved targeting capabilities.

Language: Английский

Targeting natural antioxidant polyphenols to protect neuroinflammation and neurodegenerative diseases: a comprehensive review DOI Creative Commons
Maroua Jalouli, Md. Ataur Rahman, Partha Biswas

et al.

Frontiers in Pharmacology, Journal Year: 2025, Volume and Issue: 16

Published: Jan. 24, 2025

Polyphenols, naturally occurring phytonutrients found in plant-based foods, have attracted significant attention for their potential therapeutic effects neurological diseases and neuroinflammation. These compounds possess diverse neuroprotective capabilities, including antioxidant, anti-inflammatory, anti-amyloid properties, which contribute to mitigating the progression of neurodegenerative conditions such as Alzheimer's Disease (AD), Parkinson's (PD), Dementia, Multiple Sclerosis (MS), Stroke, Huntington's (HD). Polyphenols been extensively studied ability regulate inflammatory responses by modulating activity pro-inflammatory genes influencing signal transduction pathways, thereby reducing neuroinflammation neuronal death. Additionally, polyphenols shown promise various cellular signaling pathways associated with viability, synaptic plasticity, cognitive function. Epidemiological clinical studies highlight polyphenol-rich diets decrease risk alleviate symptoms disorders Furthermore, demonstrated through regulation key Akt, Nrf2, STAT, MAPK, play critical roles neuroprotection body's immune response. This review emphasizes growing body evidence supporting combating neurodegeneration neuroinflammation, well enhancing brain health. Despite substantial promising hypotheses, further research investigations are necessary fully understand role establish them advanced targets age-related neuroinflammatory conditions.

Language: Английский

Citations

7

Interaction of starch nanoparticles with digestive enzymes and its effect on the release of polyphenols in simulated gastrointestinal fluids DOI
Jie Yang, Yujing Sun, Xuyan Dong

et al.

Food Chemistry, Journal Year: 2025, Volume and Issue: 472, P. 142883 - 142883

Published: Jan. 11, 2025

Language: Английский

Citations

0

Exploring the Mechanism of β-Cyclodextrin-Encased Phenolic Acids Functionalized with TPP for Antioxidant Activity and Targeting DOI Creative Commons
Christopher Sbarbaro, Valeria Márquez‐Miranda, Matías Leal

et al.

Antioxidants, Journal Year: 2025, Volume and Issue: 14(4), P. 465 - 465

Published: April 13, 2025

Oxidative stress on the mitochondria in a human cell is attributed to several life-risking conditions, and as such, importance of molecular structures packed with antioxidant properties structural characteristics enter help prevent such has been substantially relevant recent years. In this study, we investigated triphenylphosphonium (TPP)-conjugated phenolic acids encapsulated β-cyclodextrin (β-CD). We synthesized TPP conjugates caffeic, coumaric, cinnamic formed inclusion complexes β-CD. Our results showed successful encapsulation β-CD high efficiency. The maintained activity, slight reductions observed complexes. Furthermore, viability studies low cytotoxicity dds. Computational analyses revealed that conjugation preserved chemical reactivity acids. Molecular dynamics simulations demonstrated stable free energy calculations indicated significantly enhanced ability caffeic acid translocate across mitochondrial membranes. These highlight potential TPP-conjugated effective antioxidants improved targeting capabilities.

Language: Английский

Citations

0